Cognitive Outcomes in Trials of Two BACE Inhibitors in Alzheimer's Disease
Document Type
Article
Publication Date
10-13-2020
Publication Title
Alzheimer's and Dementia
Volume
16
Issue
11
First page number:
1483
Last page number:
1492
Abstract
Introduction: The APECS and AMARANTH trials showed that beta‐secretase (BACE) inhibitors verubecestat and lanabecestat failed to slow cognitive and functional decline in individuals with prodromal or early Alzheimer's disease. Here, the performance on secondary and exploratory cognitive measures in both studies is reported. Methods: APECS (verubecestat) and AMARANTH (lanabecestat) were randomized, double‐blind, placebo‐controlled, parallel‐group, 104‐week clinical trials conducted by different sponsors. Measures included the 3‐Domain Composite Cognition Score (CCS‐3D), Repeatable Battery for the Assessment of Neuropsychological Status (RBANS), Letter/Category Fluency, and Digit Symbol Coding. Results: Verubecestat showed worsening on the CCS‐3D Total Score, Episodic Memory, and Attention/Processing Speed domains. Lanabecestat showed worsening on the RBANS Total Score, Immediate Memory, and Visuospatial/Constructional Indexes. Both BACE inhibitors showed worsening on Digit Symbol Coding and improvements on Letter/Category Fluency. Discussion: In both studies, many measures showed treatment‐associated cognitive worsening, whereas verbal fluency tasks showed improvement.
Keywords
Alzheimer’s disease; BACE inhibition; Cognition; Lanabecestat; Verubecestat
Disciplines
Cognitive Neuroscience | Medical Neurobiology
Language
English
Repository Citation
Wessels, A. M.,
Lines, C.,
Stern, R. A.,
Kost, J.,
Voss, T.,
Mozley, L. H.,
Furtek, C.,
Mukai, Y.,
Aisen, P. S.,
Cummings, J. L.,
Tariot, P. N.,
Vellas, B.,
Dupre, N.,
Randolph, C.,
Michelson, D.,
Andersen, S. W.,
Shering, C.,
Sims, J. R.,
Egan, M. F.
(2020).
Cognitive Outcomes in Trials of Two BACE Inhibitors in Alzheimer's Disease.
Alzheimer's and Dementia, 16(11),
1483-1492.
http://dx.doi.org/10.1002/alz.12164